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Indole

Indole-related patent applications - as published by the U.S. Patent and Trademark Office (USPTO).


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NEW Simultaneous detection of off-note or boar taint related compounds in animal tissue
Teknologisk Institut
February 15, 2018 - N°20180045701

A rapid method for simultaneously quantifying the amount of compounds related to boar taint such as skatole, androstenone and indole is described. With the reduction in the number of male pigs being castrated, the number of pigs with an amount of compounds related to boar taint above a defined sensorial threshold will increase. The method for simultaneously quantifying the amount ...
NEW Blue-light-proof optical resin lens and preparation method thereof
Jiangsu Conant Optics Co., Ltd
February 15, 2018 - N°20180044505

The present invention disclose a blue-light-proof optical resin lens, comprising resin monomers, a blue light absorber and a polymerization initiator; the mass ratio of the resin monomers to the blue light absorber to the polymerization initiator is 100:0. 01-2. 00:1. 00-4. 00; the resin monomers are the mixture of allyl diglycol carbonate (adc) and polymers thereof; the blue light absorber is a benzophenone ...
NEW Ipa as a protective agent
Ixcela, Inc.
February 15, 2018 - N°20180042897

Provided is a method for reducing a potential for neurological damage of an animal at risk of head injury, by administering to the animal before exposure to the risk indole-3-propionic acid, indole lactic acid, or a salt, ester or protein complex or marginally bound preparation thereof, or a mixture thereof, in a suitable carrier.
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Inhibitors of tryptophan-2,3-dioxygenase or indoleamine-2,3-dioxygenase
Iomet Pharma Ltd.
February 08, 2018 - N°20180037553

Provided is a compound for use in medicine for inhibiting tryptophan-2,3-dioxygenase (tdo) and/or indoleamine-2,3-dioxygenase (ido), which compound comprises formula (i) wherein x1, x2, and x7, may be the same or different and each is independently selected from c and n; x3, x4, x5, and x6 may be the same or different and each is independently selected from ...
9h-pyrimido [4,5-b] indoles as bet bromodomain inhibitors
The Regents Of The University Of Michigan
February 08, 2018 - N°20180036294

The present disclosure provides substituted 9h-pyrimido [4,5-b] indoles and 5h-pyrido [4,3-b] indoles and related analogs represented by formula i and the pharmaceutically acceptable salts, hydrates, and solvates thereof, wherein r1a, w, b1, b2, g, x1, y1, y2, and y3 are as defined as set forth in the specification. The present disclosure is also directed to the use of compounds ...
Indole-based therapeutics
Colorado State University Research Foundation
February 08, 2018 - N°20180036283

Provided herein are indole-2-carboxamide compounds useful for the treatment of non-tuberculosis bacterial infections. Exemplary compounds provided herein are useful for the treatment of non-tuberculosis mycobacterial infections. Methods for preparing the indole-2-carboxamide compounds are also provided.
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Indole Patent Applications
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  • 178+ full patent PDF documents of Indole-related inventions.
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Modulators of indoleamine 2,3-dioxygenase and methods of using the same
Incyte Holdings Corporation
February 01, 2018 - N°20180030006

The present invention is directed to modulators of indoleamine 2,3-dioxygenase (ido), as well as compositions and pharmaceutical methods thereof.
Indole and indoline derivatives and methods of use thereof
January 25, 2018 - N°20180024144

Wherein a, r1, r2, r3, r4, r5, u, v, w, x, y, and z are as defined in the specification. The present application also relates to compositions comprising such compounds, and methods of treating disease conditions using such compounds and compositions, and methods for identifying such compounds.
Fused-ring compounds, pharmaceutical composition and uses thereof
Shanghai De Novo Pharmatech Co., Ltd.
January 25, 2018 - N°20180022752

This disclosure is related to a fused-ring compound of formula (i) and/or a pharmaceutically acceptable salt thereof, a pharmaceutical composition comprising the fused ring compound of formula (i) and/or a pharmaceutically acceptable salt thereof, preparation methods thereof, and use thereof in modulating activity of indoleamine 2, 3-dioxygenase (ido) and/or tryptophan 2, 3-dioxygenase (tdo). This disclosure further provides methods of ...
Compound containing indoleacetic acid core structure and use thereof
Beijing An Jian Xi Bio-medical Technology Co., Ltd.
January 25, 2018 - N°20180022700

Disclosed are a compound as shown by the following formula 1, and a pharmaceutically acceptable salt, an ester, a hydrate and an organic solvate thereof. In the formula (1), the groups r1 to r17 are independently selected from the group consisting of hydrogen, fluorine, chlorine, bromine, iodine, c1-c8 alkyl, c1-c8 alkoxy, carbonyl, hydroxyl, amino, azido, carboxyl and c1-c8 alkylsulfinyl, ...
Aryl substituted indoles and the use thereof
Purdue Pharma L.p.
January 25, 2018 - N°20180022699

The invention relates to aryl and heteroaryl substituted compounds of formula (i), and pharmaceutically acceptable salts, prodrugs, or solvates thereof, wherein g, r1, and z1-z5 are defined as set forth in the specification. The invention is also directed to the use of compounds of formula (i) to treat a disorder responsive to the blockade of sodium channels. Compounds of ...
Solid state forms of spiro-oxindole compounds
Teva Pharmaceuticals International Gmbh
January 18, 2018 - N°20180016283

The present invention provides solid state forms of certain spiro-oxindole compounds, such as funapide and the racemic mixture of funapide and its corresponding (r) enantiomer, pharmaceutical compositions comprising the solid state forms and processes for preparing the solid state forms and the pharmaceutical compositions.
Therapeutic agent for bile duct cancer
Eisai R&d Management Co., Ltd.
January 18, 2018 - N°20180015079

The present invention provides a therapeutic agent for bile duct cancer comprising 5-((2-(4-(1-(2-hydroxyethyl)piperidin-4-yl)benzamide)pyridin-4-yl)oxy)-6-(2-methoxyethoxy)-n-methyl-1h-indole-1-carboxamide or a pharmacologically acceptable salt thereof.
Indole Patent Pack
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Indole Patent Applications
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  • 178+ full patent PDF documents of Indole-related inventions.
  • Exact USPTO filing data with full-text, images, drawings & claims.
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2-oxo-1,2-dihydrobenzo[cd]indole compound and use thereof
Guangzhou Institutes Of Biomediciene And Health, Chinese Academy Of Sciences
January 11, 2018 - N°20180008574

The present invention relates to the technical field of medicinal chemistry, and in particular discloses a 2-oxo-1,2-dihydrobenzo[cd]indole compound and use thereof. The compound and pharmaceutically acceptable salt, isomer, racemate, prodrug, co-crystallized complex, hydrate, and solvate thereof can effectively inhibit the bet bromodomain receptor, and can be used for preparing a medicine for treating cancers, cell proliferative disorders, ...
Synthesis of cyclopropyl indoles and cyclohepta[b]indoles, pharmaceutical compositions containing them and method of ...
Wisconsin Alumni Research Foundation
January 04, 2018 - N°20180002318

Methods of making indole analogs using a rhodium-containing catalyst are described, along with methods of using the compounds to treat hyperglycemic, hyperlipidemic, or autoimmune disorders in mammals, and corresponding pharmaceutical compositions. Disclosed herein is a method of making indoles. The method comprises contacting a reactant of formula i wherein e is a protecting group, —so2-aryl, or —so2...
Process for preparing benzofuran-2-carboxamide derivatives
Symed Labs Limited
January 04, 2018 - N°20180002305

Provided herein are novel, commercially viable and industrially advantageous processes for the preparation of benzofuran-2-carboxamide derivatives and their intermediates, or a pharmaceutically acceptable salt thereof, in high yield and purity. Provided particularly herein are novel, commercially viable and industrially advantageous processes for the preparation of vilazodone or a pharmaceutically acceptable salt thereof in high yield and purity. Provided also ...
Diindole compounds useful in treatment of nervous system disorders
Rhode Island Board Of Education, State Of Rhode Island And Providence Plantations
January 04, 2018 - N°20180002283

The invention provides bridged diindole compounds, related pharmaceutical compositions and methods of use thereof, for the prevention, palliation and/or treatment of nervous system disorders.
Mono- or di-substituted indole derivatives as dengue viral replication inhibitors
Katholieke Universiteit Leuven
January 04, 2018 - N°20180002282

The present invention relates to mono- or di-substituted indole compounds, methods to prevent or treat dengue viral infections by using said compounds and also relates to said compounds for use as a medicine, more preferably for use as a medicine to treat or prevent dengue viral infections. The present invention furthermore relates to pharmaceutical compositions or combination preparations of the ...
[1,2,4]triazolo[1,5-a]pyridinyl substituted indole compounds
January 04, 2018 - N°20180000790

Or a salt thereof, wherein r1, r2, r3, r4, r5, m, n, and p are defined herein. Also disclosed are methods of using such compounds as inhibitors of signaling through toll-like receptor 7, or 8, or 9, and pharmaceutical compositions comprising such compounds. These compounds are useful in treating inflammatory and autoimmune diseases.
Compositions with 2,3-disubstituted indoles as charge transport materials, and display devices fabricated therefrom
Dow Global Technologies Llc
December 28, 2017 - N°20170373253

Provided is a composition comprising a compound selected from structure 1, as described herein:
Monohydroxyphenyl metabolite urine detection reagent and preparation method thereof
Jiangsu Dongbo Bio-pharmaceutical Co., Ltd.
December 28, 2017 - N°20170370853

A reagent for detection of urine monophenolic metabolites and a method for preparing the reagent are disclosed, in which the monophenolic metabolites, for example, tyrosine, p-hydroxyphenyl alanine, tryptophan and 5-hydroxyindoleacetic acid can serve as tumor markers. The reagent for detection of urine monophenolic metabolites is an aqueous solution containing nitric acid, sulfuric acid, mercuric sulfate, mercurous nitrate, nickel nitrate, phosphomolybdic ...
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